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1

Dopamine D3 Receptor Partial Agonists and Antagonists as Potential Drug Abuse Therapeutic Agents

Newman, Amy Hauck, Grundt, Peter, Nader, Michael A.

Journal:

Journal of Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 189 KB

english, 2005

2

Construction of the Steroid Framework via a Functionalized Macrocyclic Compound

Gerald Dyker, Peter Grundt

Journal:

European Journal of Organic Chemistry

Année:

1999

Langue:

english

Fichier:

PDF, 127 KB

english, 1999

3

Synthesis of Functionalized 4a-Methyl-1,2,3,4,4a,9,10,10a-octahydrophenanthrenes

Gerald Dyker, Peter Grundt

Journal:

Helvetica Chimica Acta

Année:

1999

Langue:

english

Fichier:

PDF, 120 KB

english, 1999

4

Formic Acid Catalysed Rearrangement of 5β-Methyldihydrothevinols (=3,6-Dimethoxy-5,17-dimethyl-4,5-epoxy-6,14-ethanomorphinan-7-methanols): Synthesis of New Doubly Bridged Morphinan Derivatives

David Rennison, Peter Grundt, Claire Goodyer, John W. Lewis, Stephen M. Husbands

Journal:

Chemistry & Biodiversity

Année:

2005

Langue:

english

Fichier:

PDF, 83 KB

english, 2005

5

ChemInform Abstract: Construction of the Steroid Framework via a Functionalized Macrocyclic Compound.

Gerald Dyker, Peter Grundt

Journal:

Année:

1999

Fichier:

PDF, 30 KB

1999

6

ChemInform Abstract: Synthesis of Functionalized 4a-Methyl-1,2,3,4,4a,9,10,10a-octahydrophenanthrenes.

Gerald Dyker, Peter Grundt

Journal:

Année:

1999

Fichier:

PDF, 32 KB

1999

7

ChemInform Abstract: Probes for Imidazoline Binding Sites: Synthesis and Evaluation of a Selective, Irreversible I2 Ligand.

Philippa A. Coates, Peter Grundt, Emma S. J. Robinson, David J. Nutt, Robin Tyacke, Alan L. Hudson, John W. Lewis, Stephen M. Husbands

Journal:

Année:

2000

Fichier:

PDF, 34 KB

2000

8

Dopamine D3 Receptor Partial Agonists and Antagonists as Potential Drug Abuse Therapeutic Agents

Amy Hauck Newman, Peter Grundt, Michael A. Nader

Journal:

Année:

2005

Fichier:

PDF, 8 KB

2005

9

The 14-Alkyl- and 14-Alkenyl-5β-methylindolomorphinan Series Provide δ-Selective Partial Opioid Agonists

Peter Grundt, Fernando Martinez-Bermejo, John W. Lewis, Stephen M. Husbands

Journal:

Helvetica Chimica Acta

Année:

2003

Langue:

english

Fichier:

PDF, 83 KB

english, 2003

10

Formic Acid Catalyzed Rearrangement of Thevinols (=4,5-Epoxy-3,6-dimethoxy-α,17-dimethyl-6,14-ethenomorphinan-7-methanols) and Their Vinylogous Analogues: Effects of 5β-Methyl Substitution

Peter Grundt, Fernando Martinez-Bermejo, John W. Lewis, Stephen M. Husbands

Journal:

Helvetica Chimica Acta

Année:

2003

Langue:

english

Fichier:

PDF, 198 KB

english, 2003

11

Annulated ring-systems by domino-heck-aldol-condensation and domino-Heck-Michael-addition processes

Gerald Dyker, Peter Grundt

Journal:

Tetrahedron Letters

Année:

1996

Langue:

english

Fichier:

PDF, 161 KB

english, 1996

12

Analogues of the dopamine D2 receptor antagonist L741,626: Binding, function, and SAR

Peter Grundt, Sarah Little Jane Husband, Robert R. Luedtke, Michelle Taylor, Amy Hauck Newman

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2007

Langue:

english

Fichier:

PDF, 133 KB

english, 2007

13

The effect of 6-substituted-4′,4″-difluorobenztropines on monoamine transporters and the muscarinic M1 receptor

Peter Grundt, Theresa A. Kopajtic, Jonathan L. Katz, Amy Hauck Newman

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2004

Langue:

english

Fichier:

PDF, 274 KB

english, 2004

14

Probes for imidazoline binding sites: synthesis and evaluation of a selective, irreversible I2 ligand

Philippa A. Coates, Peter Grundt, Emma S.J. Robinson, David J. Nutt, Robin Tyacke, Alan L. Hudson, John W. Lewis, Stephen M. Husbands

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2000

Langue:

english

Fichier:

PDF, 115 KB

english, 2000

15

Dopamine D3 receptor selective ligands with varying intrinsic efficacies at adenylyl cyclase inhibition and mitogenic signaling pathways

Michelle Taylor, Peter Grundt, Suzy A. Griffin, Amy Hauck Newman, Robert R. Luedtke

Journal:

Année:

2010

Langue:

english

Fichier:

PDF, 632 KB

english, 2010

16

Yawning and hypothermia in rats: effects of dopamine D3 and D2 agonists and antagonists

Gregory T. Collins, Amy Hauck Newman, Peter Grundt, Kenner C. Rice, Stephen M. Husbands, Cédric Chauvignac, Jianyong Chen, Shaomeng Wang, James H. Woods

Journal:

Psychopharmacology

Année:

2007

Langue:

english

Fichier:

PDF, 541 KB

english, 2007

17

The discriminative stimulus effects of dopamine D2- and D3-preferring agonists in rats

Mikhail N. Koffarnus, Benjamin Greedy, Stephen M. Husbands, Peter Grundt, Amy Hauck Newman, James H. Woods

Journal:

Psychopharmacology

Année:

2009

Langue:

english

Fichier:

PDF, 220 KB

english, 2009

18

Imaging brain regional and cortical laminar effects of selective D3 agonists and antagonists

Ji-Kyung Choi, Joseph B. Mandeville, Y. Iris Chen, Peter Grundt, Susanta K. Sarkar, Amy H. Newman, Bruce G. Jenkins

Journal:

Psychopharmacology

Année:

2010

Langue:

english

Fichier:

PDF, 1.13 MB

english, 2010

19

N-8-Substituted benztropinamine analogs as selective dopamine transporter ligands

Peter Grundt, Theresa A. Kopajtic, Jonathan L. Katz, Amy Hauck Newman

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2005

Langue:

english

Fichier:

PDF, 113 KB

english, 2005

20

Odontogenic lesions in opercula of permanent molars delayed in eruption

Hans Peter Philipsen, Wacharaporn Thosaporn, Peter Reichart, Gerda Grundt

Journal:

Journal of Oral Pathology & Medicine

Année:

1992

Langue:

english

Fichier:

PDF, 3.57 MB

english, 1992

21

Evaluation and initial in vitro and ex vivo characterization of the potential positron emission tomography ligand, BU99008 (2-(4,5-Dihydro-1H-imidazol-2-yl)-1- methyl-1H-indole), for the imidazoline2 binding site

Robin J. Tyacke, Amy Fisher, Emma S.J. Robinson, Peter Grundt, Emma M. Turner, Stephen M. Husbands, Alan L. Hudson, Christine A. Parker, David J. Nutt

Journal:

Année:

2012

Langue:

english

Fichier:

PDF, 830 KB

english, 2012

22

Structure–activity studies of some berberine analogs as inhibitors of Toxoplasma gondii

Bogdana Krivogorsky, Jennifer A. Pernat, Kelsi A. Douglas, Nikolas J. Czerniecki, Peter Grundt

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2012

Langue:

english

Fichier:

PDF, 172 KB

english, 2012

23

BU74, a complex oripavine derivative with potent kappa opioid receptor agonism and delayed opioid antagonism

Stephen M. Husbands, Claire L. Neilan, Jillian Broadbear, Peter Grundt, Simon Breeden, Mario D. Aceto, James H. Woods, John W. Lewis, John R. Traynor

Journal:

European Journal of Pharmacology

Année:

2005

Langue:

english

Fichier:

PDF, 164 KB

english, 2005

24

Characterization of opiates, neuroleptics, and synthetic analogs at ORL1 and opioid receptors

Nurulain Zaveri, Willma E Polgar, Cris M Olsen, Andrew B Kelson, Peter Grundt, John W Lewis, Lawrence Toll

Journal:

European Journal of Pharmacology

Année:

2001

Langue:

english

Fichier:

PDF, 139 KB

english, 2001

25

Identification of a New Scaffold for Opioid Receptor Antagonism Based on the 2-Amino-1,1-dimethyl-7-hydroxytetralin Pharmacophore

Grundt, Peter, Williams, Ian A., Lewis, John W., Husbands, Stephen M.

Journal:

Journal of Medicinal Chemistry

Année:

2004

Langue:

english

Fichier:

PDF, 116 KB

english, 2004

26

ChemInform Abstract: The Chemistry of Tryptanthrin and Its Derivatives

Ashli M. Tucker, Peter Grundt

Journal:

Année:

2012

Fichier:

PDF, 25 KB

2012

27

Direct effects of osteoprotegerin on human bone cell metabolism

Alexander Grundt, Ingo Alexander Grafe, Ute Liegibel, Ulrike Sommer, Peter Nawroth, Christian Kasperk

Journal:

Biochemical and Biophysical Research Communications

Année:

2009

Langue:

english

Fichier:

PDF, 709 KB

english, 2009

28

Evaluation of the D3 dopamine receptor selective antagonist PG01037 on l-dopa-dependent abnormal involuntary movements in rats

Rakesh Kumar, Lindsay Riddle, Suzy A. Griffin, Peter Grundt, Amy Hauck Newman, Robert R. Luedtke

Journal:

Neuropharmacology

Année:

2009

Langue:

english

Fichier:

PDF, 658 KB

english, 2009

29

Evaluation of the D3 dopamine receptor selective agonist/partial agonist PG01042 on l-dopa dependent animal involuntary movements in rats

Lindsay R. Riddle, Rakesh Kumar, Suzy A. Griffin, Peter Grundt, Amy Hauck Newman, Robert R. Luedtke

Journal:

Neuropharmacology

Année:

2011

Langue:

english

Fichier:

PDF, 646 KB

english, 2011

30

Treatment of acute edema attacks in hereditary angioedema with a bradykinin receptor-2 antagonist (Icatibant)

Bork, Konrad, Frank, Jorge, Grundt, Boris, Schlattmann, Peter, Nussberger, Juerg, Kreuz, Wolfhart

Journal:

Journal of Allergy and Clinical Immunology

Année:

2007

Langue:

english

Fichier:

PDF, 184 KB

english, 2007

31

Tryptanthrin derivatives as Toxoplasma gondii inhibitors—structure–activity-relationship of the 6-position

Krivogorsky, Bogdana, Nelson, Amber C., Douglas, Kelsi A., Grundt, Peter

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2013

Langue:

english

Fichier:

PDF, 366 KB

english, 2013

32

Novel Heterocyclic Trans Olefin Analogues of N -{4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl}arylcarboxamides as Selective Probes with High Affinity for the Dopamine D3 Receptor

Grundt, Peter, Carlson, Erin E., Cao, Jianjing, Bennett, Christina J., McElveen, Elizabeth, Taylor, Michelle, Luedtke, Robert R., Newman, Amy Hauck

Journal:

Journal of Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 217 KB

english, 2005

33

Heterocyclic Analogues of N -(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)arylcarboxamides with Functionalized Linking Chains as Novel Dopamine D3 Receptor Ligands: Potential Substance Abuse Therapeutic Agents

Grundt, Peter, Prevatt, Katherine M., Cao, Jianjing, Taylor, Michelle, Floresca, Christina Z., Choi, Ji-Kyung, Jenkins, Bruce G., Luedtke, Robert R., Newman, Amy Hauck

Journal:

Journal of Medicinal Chemistry

Année:

2007

Langue:

english

Fichier:

PDF, 427 KB

english, 2007

34

Formation of tryptanthrin compounds upon Oxone-induced dimerization of indole-3-carbaldehydes

Nelson, Amber C., Kalinowski, Emily S., Jacobson, Taylor L., Grundt, Peter

Journal:

Tetrahedron Letters

Année:

2013

Langue:

english

Fichier:

PDF, 543 KB

english, 2013

35

N -(4-(4-(2,3-Dichloro- or 2-methoxyphenyl)piperazin-1-yl)butyl)heterobiarylcarboxamides with Functionalized Linking Chains as High Affinity and Enantioselective D3 Receptor Antagonists ∥⊥

Newman, Amy Hauck, Grundt, Peter, Cyriac, George, Deschamps, Jeffrey R., Taylor, Michelle, Kumar, Rakesh, Ho, David, Luedtke, Robert R.

Journal:

Journal of Medicinal Chemistry

Année:

2009

Langue:

english

Fichier:

PDF, 317 KB

english, 2009

36

Heck Reaction and Robinson-Type Annulation: A Versatile Combination

Dyker, Gerald, Grundt, Peter, Markwitz, Hardy, Henkel, Gerald

Journal:

Journal of Organic Chemistry

Année:

1998

Langue:

english

Fichier:

PDF, 70 KB

english, 1998

37

Formation of the Decahydro(trimethylphosphine)pentaborate(1-) Anion and an Isomer of Trimethylphosphine-Pentaborane(11)

Grundt, Peter, Kodama, Goji

Journal:

Inorganic Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 1.16 MB

english, 1994

38

Opioid Binding and in Vitro Profiles of a Series of 4-Hydroxy-3-methoxyindolomorphinans. Transformation of a δ-Selective Ligand into a High Affinity κ-Selective Ligand by Introduction of a 5,14-Substituted Bridge

Grundt, Peter, Martinez-Bermejo, Fernando, Lewis, John W., Husbands, Stephen M.

Journal:

Journal of Medicinal Chemistry

Année:

2003

Langue:

english

Fichier:

PDF, 69 KB

english, 2003

39

Guanidino N-Substituted and N,N-Disubstituted Derivatives of the κ-Opioid Antagonist GNTI

Black, Shannon L., Chauvignac, Cedric, Grundt, Peter, Miller, Carl N., Wood, Susan, Traynor, John R., Lewis, John W., Husbands, Stephen M.

Journal:

Journal of Medicinal Chemistry

Année:

2003

Langue:

english

Fichier:

PDF, 110 KB

english, 2003

40

Structure−Activity Relationships at Monoamine Transporters for a Series of N-Substituted 3α-(Bis[4-fluorophenyl]methoxy)tropanes: Comparative Molecular Field Analysis, Synthesis, and Pharmacological Evaluation

Kulkarni, Santosh S., Grundt, Peter, Kopajtic, Theresa, Katz, Jonathan L., Newman, Amy Hauck

Journal:

Journal of Medicinal Chemistry

Année:

2004

Langue:

english

Fichier:

PDF, 237 KB

english, 2004

41

7,9-Dichloro-6 H ,12 H -indolo[2,1- b ]quinazoline-6,12-dione

Grundt, Peter, Douglas, Kelsi A., Krivogorsky, Bogdana, Nemykin, Victor N.

Journal:

Acta Crystallographica Section E Structure Reports Online

Année:

2010

Langue:

english

Fichier:

PDF, 562 KB

english, 2010

42

9- O -Ethylberberrubinium iodide monohydrate

Grundt, Peter, Pernat, Jennifer, Krivogorsky, Bogdana, Halverson, Melanie A., Berry, Steven M.

Journal:

Acta Crystallographica Section E Structure Reports Online

Année:

2010

Langue:

english

Fichier:

PDF, 906 KB

english, 2010

43

rac -(6 S )-6-Hydroxy-6-{2-[2-(propan-2-ylidene)hydrazinylidene]propyl}indolo[2,1- b ]quinazolin-12(6 H )-one

Rodstein, Matthew E., Steffen, Paul D., Krivogorsky, Bogdana, Grundt, Peter

Journal:

Acta Crystallographica Section E Structure Reports Online

Année:

2011

Langue:

english

Fichier:

PDF, 834 KB

english, 2011

44

14-Amino, 14-Alkylamino, and 14-Acylamino Analogs of Oxymorphindole. Differential Effects on Opioid Receptor Binding and Functional Profiles

Grundt, Peter, Jales, Andrew R., Traynor, John R., Lewis, John W., Husbands, Stephen M.

Journal:

Journal of Medicinal Chemistry

Année:

2003

Langue:

english

Fichier:

PDF, 65 KB

english, 2003

45

ChemInform Abstract: Formation of Tryptanthrin Compounds upon Oxone-Induced Dimerization of Indole-3-carbaldehydes.

Nelson, Amber C., Kalinowski, Emily S., Jacobson, Taylor L., Grundt, Peter

Journal:

Année:

2014

Fichier:

PDF, 23 KB

2014

46

ChemInform Abstract: Is the 2,3-Carbon-Carbon Bond of Indole Really Inert to Oxidative Cleavage by Oxone? - Synthesis of Isatoic Anhydrides from Indoles.

Nelson, Amber C., Kalinowski, Emily S., Czerniecki, Nikolas J., Jacobson, Taylor L., Grundt, Peter

Journal:

Année:

2014

Fichier:

PDF, 26 KB

2014

47

Effects of selective dopaminergic compounds on a delay-discounting task

Koffarnus, Mikhail N., Newman, Amy H., Grundt, Peter, Rice, Kenner C., Woods, James H.

Journal:

Behavioural Pharmacology

Année:

2011

Langue:

english

Fichier:

PDF, 321 KB

english, 2011

48

Yawning and locomotor behavior induced by dopamine receptor agonists in mice and rats

Li, Su-Min, Collins, Gregory T., Paul, Noel M., Grundt, Peter, Newman, Amy H., Xu, Ming, Grandy, David K., Woods, James H., Katz, Jonathan L.

Journal:

Behavioural Pharmacology

Année:

2010

Langue:

english

Fichier:

PDF, 301 KB

english, 2010

49

Cocaine self-administration in dopamine D₃ receptor knockout mice.

Caine, S. Barak, Thomsen, Morgane, Barrett, Andrew C., Collins, Gregory T., Grundt, Peter, Newman, Amy Hauck, Butler, Paul, Xu, Ming

Journal:

Experimental and Clinical Psychopharmacology

Année:

2012

Langue:

english

Fichier:

PDF, 242 KB

english, 2012

50

Rapid susceptibility testing of multi-drug resistant Escherichia coli and Klebsiella by glucose metabolization monitoring

Kittel, Maximilian, Findeisen, Peter, Ghebremedhin, Beniam, Miethke, Thomas, Grundt, Alexander, Ahmad-Nejad, Parviz, Neumaier, Michael

Journal:

Clinical Chemistry and Laboratory Medicine

Année:

2019

Langue:

english

Fichier:

PDF, 623 KB

english, 2019